Acute Porphyria Drug Database

Monograph

G04BE08 - Tadalafil
Propably not porphyrinogenic
PNP

Rationale
Substrate for CYP 3A4. Does not give rise to CYP induction.
Chemical description
Used (tablets 10-20 mg/dose) in erectile dysfunction. Selective inhibitor of cGMP- specific fhosphodiesterase, giving rise to relaxation of smooth muscle and increased blood flow into penis. Mainly metabolized by CYP 3A4.
Similar drugs
Explore alternative drugs in similar therapeutic classes G04B / G04BE or go back.
Tradenames
This list comprises raw data collected from different countries. In some cases, a more comprehensive list of available drug packages is included. Consequently, very similar terms may therefore appear multiple times. Bold names are the searchable terms, while the gray names that follow are all mapped to the bolded term.
Note: The cleaning is done automatically by a proprietary algorithm, and it may produce errors. We strive to improve it continuously.


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